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Contents Volume 79 (2002)
Journal of Controlled Release 79 (2002) 315–316 www.elsevier.com / locate / jconrel
Contents Volume 79 (2002) Vol. 79, Nos. 1 – 3 (19 FEBRUARY 2002)
Rapid communication A cationic sub-micron emulsion (MF59 / DOTAP) is an effective delivery system for DNA vaccines G. Ott, M. Singh, J. Kazzaz, M. Briones, E. Soenawan, M. Ugozzoli, D.T. O’ Hagan ( Emeryville, CA, USA) Reviews Formulation aspects in the development of osmotically controlled oral drug delivery systems R.K. Verma, D.M. Krishna, S. Garg ( Punjab, India) Targeting to macrophages: role of physicochemical properties of particulate carriers—liposomes and microspheres—on the phagocytosis by macrophages ´ (Amarillo, TX, USA, Madrid, Spain) F. Ahsan, I.P. Rivas, M. A. Khan, A.I. Torres Suarez Research papers Anticancer drug delivery systems: N 4 -acyl poly(ethyleneglycol) prodrugs of ara-C. I. Efficacy in solid tumors Y.H. Choe, C.D. Conover, D. Wu, M. Royzen, R.B. Greenwald ( Piscataway, NJ, USA) Anticancer drug delivery systems: multi-loaded N 4 -acyl poly(ethylene glycol) prodrugs of ara-C. II. Efficacy in ascites and solid tumors Y.H. Choe, C.D. Conover, D. Wu, M. Royzen, Y. Gervacio, V. Borowski, M. Mehlig, R.B. Greenwald ( Piscataway, NJ, USA) A floating-type oral dosage form for piroxicam based on hollow polycarbonate microspheres: in vitro and in vivo evaluation in rabbits N. J. Joseph, S. Lakshmi, A. Jayakrishnan ( Trivandrum, India) A novel sustained-release formulation of insulin with dramatic reduction in initial rapid release M. Takenaga, Y. Yamaguchi, A. Kitagawa, Y. Ogawa, Y. Mizushima, R. Igarashi ( Kawasaki, Japan) Transdermal drug delivery of imipramine hydrochloride. I. Effect of terpenes A.K. Jain, N.S. Thomas, R. Panchagnula ( Punjab, India) Colon-specific delivery of prednisolone-appended a-cyclodextrin conjugate: alleviation of systemic side effect after oral administration H. Yano, F. Hirayama, M. Kamada, H. Arima, K. Uekama ( Kumamoto, Japan) Percutaneous penetration and skin metabolism of ethylsalicylate-containing agent, TU-2100: in-vitro and in-vivo evaluation in guinea pigs A.C. Sintov, C. Behar-Canetti, Y. Friedman, D. Tamarkin ( Beer Sheva, Rehovot, Israel) PLGA–mPEG nanoparticles of cisplatin: in vitro nanoparticle degradation, in vitro drug release and in vivo drug residence in blood properties K. Avgoustakis, A. Beletsi, Z. Panagi, P. Klepetsanis, A.G. Karydas, D.S. Ithakissios ( Rion, Athens, Greece) Assessment of protein release kinetics, stability and protein polymer interaction of lysozyme encapsulated poly( D,L-lactide-co-glycolide) microspheres G. Jiang, B.H. Woo, F. Kang, J. Singh, P.P. DeLuca ( Lexington, KY, Fargo, ND, USA) The enhancing effect of nasal absorption of FITC-dextran 4,400 by b-sitosterol b-D-glucoside in rabbits K. Nakamura, Y. Maitani, K. Takayama ( Tokyo, Japan)
PII: S0168-3659( 02 )00014-7
1
7
29
41
55
71 81 93
103
113
123
137 147
316
Contents Volume 79 (2002)
Modulation of active pharmaceutical material release from a novel ‘tablet in capsule system’ containing an effervescent blend M.C. Gohel, M. Sumitra G ( Gujarat, India) The effect of fatty acid substitution on the in vitro release of amphotericin B from micelles composed of poly(ethylene oxide)-block-poly(N-hexyl stearate-L-aspartamide) A. Lavasanifar, J. Samuel, G.S. Kwon ( Edmonton, Canada, Madison, WI, USA) Ex vivo bioadhesion and in vivo testosterone bioavailability study of different bioadhesive formulations based on starch-g-poly(acrylic acid) copolymers and starch / poly(acrylic acid) mixtures D. Ameye, J. Voorspoels, P. Foreman, J. Tsai, P. Richardson, S. Geresh, J.P. Remon ( Gent, Belgium, Bridgewater, NJ, USA, Beer-Sheva, Israel) Lectin-mediated drug delivery: influence of mucin on cytoadhesion of plant lectins in vitro M. Wirth, K. Gerhardt, C. Wurm, F. Gabor ( Vienna, Austria) Double emulsions: how does release occur? K. Pays, J. Giermanska-Kahn, B. Pouligny, J. Bibette, F. Leal-Calderon ( Pessac, Paris, France) Sustained-delivery of an apolipoproteinE–peptidomimetic using multivesicular liposomes lowers serum cholesterol levels M.P. Ramprasad, G.M. Anantharamaiah, D.W. Garber, N.V. Katre ( San Diego, CA, Birmingham, AL, USA) In vivo assessment of skin electroporation using square wave pulses ´ ( Brussels, Belgium, Archamps, France) N. Dujardin, E. Staes, Y. Kalia, P. Clarys, R. Guy, V. Preat Enhanced tumor cell selectivity of adriamycin-monoclonal antibody conjugate via a poly(ethylene glycol)-based cleavable linker T. Suzawa, S. Nagamura, H. Saito, S. Ohta, N. Hanai, J. Kanazawa, M. Okabe, M. Yamasaki ( Tokyo, Shizuoka, Japan) Development of a novel nasal nicotine formulation comprising an optimal pulsatile and sustained plasma nicotine profile for smoking cessation Yu.-H. Cheng, P. Watts, M. Hinchcliffe, R. Hotchkiss, R. Nankervis, N.F. Faraj, A. Smith, S.S. Davis, L. Illum ( Nottingham, UK) Gene delivery Optimization of factors influencing the transfection efficiency of folate–PEG–folate-graft-polyethylenimine J.M. Benns, R.I. Mahato, S.W. Kim ( Salt Lake City, UT, USA) A new synthesis of galactose-poly(ethylene glycol)-polyethylenimine for gene delivery to hepatocytes K. Sagara, S.W. Kim ( Salt Lake City, UT, USA) PEG grafted polylysine with fusogenic peptide for gene delivery: high transfection efficiency with low cytotoxicity H. Lee, J.H. Jeong, T.G. Park ( Taejon, South Korea) Notes Multipulse drug permeation across a membrane driven by a chemical pH-oscillator G.P. Misra, R. A. Siegel ( Minneapolis, MN, USA) Chemical hydrolysis of DOTAP and DOPE in a liposomal environment E. A. A.M. Vernooij, J. J. Kettenes-van den Bosch, W. J.M. Underberg, D. J. A. Crommelin ( Utrecht, Leiden, The Netherlands) Calendar of Events Author Index Volume 79 Subject Index Volume 79 Contents Volume 79
157
165
173 183 193
207 219
229
243
255 271 283
293
299 305 309 313 315
Contents Volume 79 (2002) Vol. 79, Nos. 1 – 3 (19 FEBRUARY 2002)
Rapid communication A cationic sub-micron emulsion (MF59 / DOTAP) is an effective delivery system for DNA vaccines G. Ott, M. Singh, J. Kazzaz, M. Briones, E. Soenawan, M. Ugozzoli, D.T. O’ Hagan ( Emeryville, CA, USA) Reviews Formulation aspects in the development of osmotically controlled oral drug delivery systems R.K. Verma, D.M. Krishna, S. Garg ( Punjab, India) Targeting to macrophages: role of physicochemical properties of particulate carriers—liposomes and microspheres—on the phagocytosis by macrophages ´ (Amarillo, TX, USA, Madrid, Spain) F. Ahsan, I.P. Rivas, M. A. Khan, A.I. Torres Suarez Research papers Anticancer drug delivery systems: N 4 -acyl poly(ethyleneglycol) prodrugs of ara-C. I. Efficacy in solid tumors Y.H. Choe, C.D. Conover, D. Wu, M. Royzen, R.B. Greenwald ( Piscataway, NJ, USA) Anticancer drug delivery systems: multi-loaded N 4 -acyl poly(ethylene glycol) prodrugs of ara-C. II. Efficacy in ascites and solid tumors Y.H. Choe, C.D. Conover, D. Wu, M. Royzen, Y. Gervacio, V. Borowski, M. Mehlig, R.B. Greenwald ( Piscataway, NJ, USA) A floating-type oral dosage form for piroxicam based on hollow polycarbonate microspheres: in vitro and in vivo evaluation in rabbits N. J. Joseph, S. Lakshmi, A. Jayakrishnan ( Trivandrum, India) A novel sustained-release formulation of insulin with dramatic reduction in initial rapid release M. Takenaga, Y. Yamaguchi, A. Kitagawa, Y. Ogawa, Y. Mizushima, R. Igarashi ( Kawasaki, Japan) Transdermal drug delivery of imipramine hydrochloride. I. Effect of terpenes A.K. Jain, N.S. Thomas, R. Panchagnula ( Punjab, India) Colon-specific delivery of prednisolone-appended a-cyclodextrin conjugate: alleviation of systemic side effect after oral administration H. Yano, F. Hirayama, M. Kamada, H. Arima, K. Uekama ( Kumamoto, Japan) Percutaneous penetration and skin metabolism of ethylsalicylate-containing agent, TU-2100: in-vitro and in-vivo evaluation in guinea pigs A.C. Sintov, C. Behar-Canetti, Y. Friedman, D. Tamarkin ( Beer Sheva, Rehovot, Israel) PLGA–mPEG nanoparticles of cisplatin: in vitro nanoparticle degradation, in vitro drug release and in vivo drug residence in blood properties K. Avgoustakis, A. Beletsi, Z. Panagi, P. Klepetsanis, A.G. Karydas, D.S. Ithakissios ( Rion, Athens, Greece) Assessment of protein release kinetics, stability and protein polymer interaction of lysozyme encapsulated poly( D,L-lactide-co-glycolide) microspheres G. Jiang, B.H. Woo, F. Kang, J. Singh, P.P. DeLuca ( Lexington, KY, Fargo, ND, USA) The enhancing effect of nasal absorption of FITC-dextran 4,400 by b-sitosterol b-D-glucoside in rabbits K. Nakamura, Y. Maitani, K. Takayama ( Tokyo, Japan)
PII: S0168-3659( 02 )00014-7
1
7
29
41
55
71 81 93
103
113
123
137 147
316
Contents Volume 79 (2002)
Modulation of active pharmaceutical material release from a novel ‘tablet in capsule system’ containing an effervescent blend M.C. Gohel, M. Sumitra G ( Gujarat, India) The effect of fatty acid substitution on the in vitro release of amphotericin B from micelles composed of poly(ethylene oxide)-block-poly(N-hexyl stearate-L-aspartamide) A. Lavasanifar, J. Samuel, G.S. Kwon ( Edmonton, Canada, Madison, WI, USA) Ex vivo bioadhesion and in vivo testosterone bioavailability study of different bioadhesive formulations based on starch-g-poly(acrylic acid) copolymers and starch / poly(acrylic acid) mixtures D. Ameye, J. Voorspoels, P. Foreman, J. Tsai, P. Richardson, S. Geresh, J.P. Remon ( Gent, Belgium, Bridgewater, NJ, USA, Beer-Sheva, Israel) Lectin-mediated drug delivery: influence of mucin on cytoadhesion of plant lectins in vitro M. Wirth, K. Gerhardt, C. Wurm, F. Gabor ( Vienna, Austria) Double emulsions: how does release occur? K. Pays, J. Giermanska-Kahn, B. Pouligny, J. Bibette, F. Leal-Calderon ( Pessac, Paris, France) Sustained-delivery of an apolipoproteinE–peptidomimetic using multivesicular liposomes lowers serum cholesterol levels M.P. Ramprasad, G.M. Anantharamaiah, D.W. Garber, N.V. Katre ( San Diego, CA, Birmingham, AL, USA) In vivo assessment of skin electroporation using square wave pulses ´ ( Brussels, Belgium, Archamps, France) N. Dujardin, E. Staes, Y. Kalia, P. Clarys, R. Guy, V. Preat Enhanced tumor cell selectivity of adriamycin-monoclonal antibody conjugate via a poly(ethylene glycol)-based cleavable linker T. Suzawa, S. Nagamura, H. Saito, S. Ohta, N. Hanai, J. Kanazawa, M. Okabe, M. Yamasaki ( Tokyo, Shizuoka, Japan) Development of a novel nasal nicotine formulation comprising an optimal pulsatile and sustained plasma nicotine profile for smoking cessation Yu.-H. Cheng, P. Watts, M. Hinchcliffe, R. Hotchkiss, R. Nankervis, N.F. Faraj, A. Smith, S.S. Davis, L. Illum ( Nottingham, UK) Gene delivery Optimization of factors influencing the transfection efficiency of folate–PEG–folate-graft-polyethylenimine J.M. Benns, R.I. Mahato, S.W. Kim ( Salt Lake City, UT, USA) A new synthesis of galactose-poly(ethylene glycol)-polyethylenimine for gene delivery to hepatocytes K. Sagara, S.W. Kim ( Salt Lake City, UT, USA) PEG grafted polylysine with fusogenic peptide for gene delivery: high transfection efficiency with low cytotoxicity H. Lee, J.H. Jeong, T.G. Park ( Taejon, South Korea) Notes Multipulse drug permeation across a membrane driven by a chemical pH-oscillator G.P. Misra, R. A. Siegel ( Minneapolis, MN, USA) Chemical hydrolysis of DOTAP and DOPE in a liposomal environment E. A. A.M. Vernooij, J. J. Kettenes-van den Bosch, W. J.M. Underberg, D. J. A. Crommelin ( Utrecht, Leiden, The Netherlands) Calendar of Events Author Index Volume 79 Subject Index Volume 79 Contents Volume 79
157
165
173 183 193
207 219
229
243
255 271 283
293
299 305 309 313 315