Contents to Vol. 23

European Journal of Pharmaceutical Sciences 23 (2004) 413–415

Contents, Volume 23 Vol. 23/1, September 2004 Reviews Allosteric modulation of neurotransmitter transporters at excitatory synapses R.J. Vandenberg, P. Ju, K.R. Aubrey, R.M. Ryan, A.D. Mitrovic

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Drug permeation in biomembranes. In vitro and in silico prediction and influence of physicochemical properties A. Ma¨lkia¨, L. Murtoma¨ki, A. Urtti, K. Kontturi

13

Research papers Oesophageal bioadhesion of sodium alginate suspensions: particle swelling and mucosal retention J.C. Richardson, P.W. Dettmar, F.C. Hampson, C.D. Melia

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Improvement of gliquidone hypoglycaemic effect in rats by cyclodextrin formulations A. Miro, F. Quaglia, U. Sorrentino, M.I. La Rotonda, R. D’Emmanuele Di Villa Bianca, R. Sorrentino

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Physicochemical studies on the stability of influenza haemagglutinin in vaccine bulk material D.M.A.M. Luykx, M.G. Casteleijn, W. Jiskoot, J. Westdijk, P.M.J.M. Jongen

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Effect of different sterilisation methods on the properties of bioadhesive powders and ocular minitablets, and clinical evaluation W. Weyenberg, A. Vermeire, E. D’Haese, G. Vanhaelewyn, P. Kestelyn, F. Callens, H.J. Nelis, J.P. Remon, A. Ludwig

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Imidazole H3-antagonists: relationship between structure and ex vivo binding to rat brain H3-receptors F. Vacondio, M. Mor, C. Silva, V. Zuliani, M. Rivara, S. Rivara, F. Bordi, P.V. Plazzi, F. Magnanini, S. Bertoni, V. Ballabeni, E. Barocelli, P.-A. Carrupt, B. Testa

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Role of excipients in hydrate formation kinetics of theophylline in wet masses studied by near-infrared spectroscopy A.C. Jørgensen, S. Airaksinen, M. Karjalainen, P. Luukkonen, J. Rantanen, J. Yliruusi

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Calendar of Events

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Instructions to Authors

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Vol. 23/2, October 2004 Research papers Microspectroscopic FT-IR mapping system as a tool to assess blend homogeneity of drug–excipient mixtures T.-H. Lee, S.-Y. Lin

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Evolution of the interaction of a new chemical entity, eflucimibe, with g-cyclodextrin during kneading process A. Gil, A. Chamayou, E. Leverd, J. Bougaret, M. Baron, G. Couarraze

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Photophysicals and photochemicals studies of zinc(II) phthalocyanine in long time circulation micelles for Photodynamic Therapy use M.N. Sibata, A.C. Tedesco, J.M. Marchetti

131

The role of particle engineering in relation to formulation and de-agglomeration principle in the development of a dry powder formulation for inhalation of cetrorelix G.S. Zijlstra, W.L.J. Hinrichs, A.H. de Boer, H.W. Frijlink

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doi:10.1016/S0928-0987(04)00275-1

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Contents, Volume 23 (2004) 413–415

Design, synthesis and in vitro evaluation of novel water-soluble prodrugs of buparvaquone A. Ma¨ntyla¨, J. Rautio, T. Nevalainen, P. Keski-Rahkonen, J. Vepsa¨lainen, T. Ja¨rvinen

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Preparation of budesonide– and indomethacin–hydroxypropyl-b-cyclodextrin (HPBCD) complexes using a single-step, organic-solvent-free supercritical fluid process N. Bandi, W. Wei, C.B. Roberts, L.P. Kotra, U.B. Kompella

159

The effect of vessel material on granules produced in a high-shear mixer A.M. Bouwman, M.R. Visser, A.C. Eissens, J.A. Wesselingh, H.W. Frijlink

169

Substrates and inhibitors of efflux proteins interfere with the MTT assay in cells and may lead to underestimation of drug toxicity K.-S. Vellonen, P. Honkakoski, A. Urtti

181

Impact of serum on clearance predictions obtained from suspensions and primary cultures of rat hepatocytes N. Blanchard, L. Richert, B. Notter, F. Delobel, P. David, P. Coassolo, T. Lave´

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EUFEPS Announcement

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Calendar of Events

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Vol. 23/3, November 2004 Research papers Tertiary selenoamide compounds are useful superoxide radical scavengers in vitro H. Takahashi, A. Nishina, H. Kimura, K. Motoki, M. Koketsu, H. Ishihara

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Pharmacokinetics of levosimendan and its active metabolite OR-1896 in rapid and slow acetylators S. Antila, U. Pesonen, L. Lehtonen, P. Tapanainen, H. Nikkanen, K. Vaahtera, H. Scheinin

213

Permeability through DOPC/dodecane membranes: measurement and LFER modelling F.T.T. Huque, K. Box, J.A. Platts, J. Comer

223

Comparison of cannabinoid ligands affinities and efficacies in murine tissues and in transfected cells expressing human recombinant cannabinoid receptors S.J. Govaerts, E. Hermans, D.M. Lambert

233

Albumin loaded microsphere of amphiphilic poly(ethylene glycol)/poly(a-ester) multiblock copolymer J.-H. Kim, Y.H. Bae

245

A concentric cylinder shear device for the study of stability in intravenous emulsions J. Han, C. Washington, C.D. Melia

253

The characteristics of spontaneously forming physically cross-linked hydrogels composed of two water-soluble phospholipid polymers for oral drug delivery carrier I: hydrogel dissolution and insulin release under neutral pH condition K. Nam, J. Watanabe, K. Ishihara

261

Choice of rotation speed (rpm) for bio-relevant drug dissolution testing using a crescent-shaped spindle S.A. Qureshi

271

Isoproterenol-induced myocardial infarction in rabbits. Protection by propranolol or labetalol: a proposed non-invasive procedure A. Pinelli, S. Trivulzio, L. Tomasoni, S. Brenna, E. Bonacina, R. Accinni

277

Solubilisation of poorly water-soluble drugs during in vitro lipolysis of medium- and long-chain triacylglycerols J.Ø. Christensen, K. Schultz, B. Mollgaard, H.G. Kristensen, A. Mullertz

287

Calendar

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Contents, Volume 23 (2004) 413–415

415

Vol. 23/4–5, December 2004 Review Functional consequences of 7TM receptor dimerization J.L. Hansen, S.P. Sheikh

301

Research papers Acyclovir prodrug for the intestinal di/tri-peptide transporter PEPT1: comparison of in vivo bioavailability in rats and transport in Caco-2 cells A.E. Thomsen, M.S. Christensen, M.A. Bagger, B. Steffansen

319

Development of a novel approach towards predicting the milling behaviour of pharmaceutical powders C.C. Kwan, Y.Q. Chen, Y.L. Ding, D.G. Papadopoulos, A.C. Bentham, M. Ghadiri

327

4

N -alkyloxycarbonyl derivatives of cytosine: physicochemical characterisation, and cytosine regeneration rates and release from alginic acid gels K. Petersson, B.T. Pedersen, D. Stærk, K.A. Krogfelt, C. Larsen

337

Preparation of ibuprofen-loaded liquid suppository using eutectic mixture system with menthol C.S. Yong, Y.-K. Oh, S.H. Jung, J.-D. Rhee, H.-D. Kim, C.-K. Kim, H.-G. Choi

347

Development and validation of a direct, non-destructive quantitative method for medroxyprogesterone acetate in a pharmaceutical suspension using FT-Raman spectroscopy T.R.M. De Beer, G.J. Vergote, W.R.G. Baeyens, J.P. Remon, C. Vervaet, F. Verpoort

355

New optimized piperamide analogues with potent in vivo hypotensive properties C.M Duarte, H. Verli, J.X. de Arau´jo-Ju´nior, I.A. de Medeiros, E.J. Barreiro, C.A.M. Fraga

363

Electrochemical and calorimetric study of oligonucleotide complexation with cetylpyridinium chloride S. Hakkarainen, A.-K. Kontturi, K. Kontturi, A. Urtti

371

Improvement of warfarin biopharmaceutics by conjugation with poly(ethylene glycol) M. Zacchigna, G. Di Luca, F. Cateni, V. Maurich

379

Localisation of drug permeability along the rat small intestine, using markers of the paracellular, transcellular and some transporter routes O. Lacombe, J. Woodley, C. Solleux, J.-M. Delbos, C. Boursier-Neyret, G. Houin

385

A novel method for coupling doxorubicin to lactosaminated human albumin by an acid sensitive hydrazone bond: synthesis, characterization and preliminary biological properties of the conjugate G. Di Stefano, M. Lanza, F. Kratz, L. Merina, L. Fiume

393

EUFEPS Membership Form

399

EJPS Individual Subscription Form

400

EUFEPS Announcement

401

Calendar of Events

405

Author Index Vol. 23

409

Contents Vol. 23

413