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Contents to Vol. 25
European Journal of Pharmaceutical Sciences 25 (2005) 479–482
Contents, Volume 25 Vol. 25/1, May 2005 Review Microdialysis—theoretical background and recent implementation in applied life-sciences N. Plock, C. Kloft
1
Research papers Pharmacodynamic behaviour of the selective cyclooxygenase-2 inhibitor lumiracoxib in the lipopolysaccharidestimulated rat air pouch model R.E. Esser, R. Miserendino-Molteni, M. Sharr, X. Zhang, W. Porter, L. Ramos, J.A. Cramer, S. Zhuang, A. Georgieva, W. Maniara
25
Chitosan-reinforced alginate microspheres obtained through the emulsification/internal gelation technique A.J. Ribeiro, C. Silva, D. Ferreira, F. Veiga
31
Melt sonocrystallization of ibuprofen: Effect on crystal properties M. Manish, J. Harshal, P. Anant
41
Characterization of the 13-cis-retinoic acid/cyclodextrin inclusion complexes by phase solubility, photostability, physicochemical and computational analysis K.L. Yap, X. Liu, J.C. Thenmozhiyal, P.C. Ho
49
Vanillin suppresses in vitro invasion and in vivo metastasis of mouse breast cancer cells K. Lirdprapamongkol, H. Sakurai, N. Kawasaki, M.-K. Choo, Y. Saitoh, Y. Aozuka, P. Singhirunnusorn, S. Ruchirawat, J. Svasti, I. Saiki
57
A new sunscreen of the cinnamate class: Synthesis and enzymatic hydrolysis evaluation of glyceryl esters of p-methoxycinnamic acid Z.M.F. de Freitas, E.P. dos Santos, J.F. da Rocha, G.M. Dellamora-Ortiz, J.C.S. Gonçalves
67
Characterization of the rotating dialysis cell as an in vitro model potentially useful for simulation of the pharmacokinetic fate of intra-articularly administered drugs B.T. Pedersen, J. Østergaard, S.W. Larsen, C. Larsen
73
Atomic force microscopy and photon correlation spectroscopy: Two techniques for rapid characterization of liposomes B. Ruozi, G. Tosi, F. Forni, M. Fresta, M.A. Vandelli
81
Tissue distribution, pharmacokinetics and identification of roscovitine metabolites in rat M. Vita, M. Abdel-Rehim, S. Olofsson, Z. Hassan, L. Meurling, Å. Sidén, M. Sidén, T. Pettersson, M. Hassan
91
A solid-state NMR study of molecular mobility and phase separation in co-spray-dried protein–sugar particles E.J. Suihko, R.T. Forbes, D.C. Apperley
105
Permeability of pig urinary bladder wall: the effect of chitosan and the role of calcium M. Kerec, M. Bogataj, P. Veranicˇ , A. Mrhar
113
Estimation of dosing strategies aiming at maximizing utility or responder probability, using oxybutynin as an example drug S. Jönsson, M.O. Karlsson
123
doi:10.1016/S0928-0987(05)00185-5
480
Contents, Volume 25 (2005) 479–482
A comparative study of the potential of solid triglyceride nanostructures coated with chitosan or poly(ethylene glycol) as carriers for oral calcitonin delivery M. Garcia-Fuentes, C. Prego, D. Torres, M.J. Alonso
133
Pyrimidine and nucleoside -esters of L-Glu-Sar: Synthesis, stability and interaction with hPEPT1 A.H. Eriksson, P.L. Elm, M. Begtrup, B. Brodin, R. Nielsen, B. Steffansen
145
A simple method for differentiation of monoisotopic drug metabolites with hydrogen–deuterium exchange liquid chromatography/electrospray mass spectrometry A. Tolonen, M. Turpeinen, J. Uusitalo, O. Pelkonen
155
Pharmacokinetic–pharmacodynamic modelling of the schedule-dependent effect of the anti-cancer agent CHS 828 in a rat hollow fibre model L.E. Friberg, S.B. Hassan, E. Lindhagen, R. Larsson, M.O. Karlsson
163
EUFEPS Announcement
175
Calendar of Events
179
Instructions to Authors
183
Vol. 25/2–3, June 2005 Research papers Effect of experimental pH on the in vitro permeability in intact rabbit intestines and Caco-2 monolayer K.-J. Lee, N. Johnson, J. Castelo, P.J. Sinko, G. Grass, K. Holme, Y.-H. Lee
193
[99mTc]-hexakis-2-methoxyisobutyl
Biphasic accumulation kinetics of isonitrile in tumour cells and its modulation by lipophilic P-glycoprotein ligands T. Márián, L. Balkay, G. Szabó, Z.T. Krasznai, Z. Hernádi, L. Galuska, J. Szabó-Péli, O. Ésik, L. Trón, Z. Krasznai
201
pH-Dependent passive and active transport of acidic drugs across Caco-2 cell monolayers S. Neuhoff, A.-L. Ungell, I. Zamora, P. Artursson
211
Effect of staurosporine on N-glycosylation and cell adhesion to fibronectin of SW480 human colorectal adenocarcinoma cells T. Sato, M. Takahashi, T. Kawado, E. Takayama, K. Furukawa
221
AZD3582 increases heme oxygenase-1 expression and antioxidant activity in vascular endothelial and gastric mucosal cells G. Berndt, N. Grosser, J. Hoogstraate, H. Schröder
229
SDS-aided immobilization and controlled release of camptothecin from agarose hydrogel J. Liu, L. Li
237
QSAR analysis of substituted bis[(acridine-4-carboxamide)propyl]methylamines using optimized block-wise variable combination by particle swarm optimization for partial least squares modeling L. Lin, W.-Q. Lin, J.-H. Jiang, G.-L. Shen, R.-Q. Yu
245
Synthesis and antiamoebic activity of 3,7-dimethyl-pyrazolo[3,4-e][1,2,4] triazin-4-yl thiosemicarbazide derivatives S. Singh, K. Husain, F. Athar, A. Azam
255
Modulation of drug transport by selected flavonoids: Involvement of P-gp and OCT? M. Ofer, S. Wolffram, A. Koggel, H. Spahn-Langguth, P. Langguth
263
Acid–base properties of selected flavonoid glycosides C. Mielczarek
273
Polyelectrolyte complex formation and stability when mixing polyanions and polycations in salted media: A model study related to the case of body fluids T. Etrych, L. Leclercq, M. Boustta, M. Vert
281
Contents, Volume 25 (2005) 479–482
481
State of insulin self-association does not affect its absorption from the pulmonary route A. Hussain, F. Ahsan
289
Targeting liposomes with protein drugs to the blood–brain barrier in vitro C.C. Visser, S. Stevanovic´, L.H. Voorwinden, L. van Bloois, P.J. Gaillard, M. Danhof, D.J.A. Crommelin, A.G. de Boer
299
Investigation of the enhancing mechanism of sodium N-[8-(2-hydroxybenzoyl)amino]caprylate effect on the intestinal permeability of polar molecules utilizing a voltage clamp method S. Hess, V. Rotshild, A. Hoffman
307
Physical stability of the amorphous state of loperamide and two fragment molecules in solid dispersions with the polymers PVP-K30 and PVP-VA64 I. Weuts, D. Kempen, A. Decorte, G. Verreck, J. Peeters, M. Brewster, G. Van den Mooter
313
Hydrophilic solutes in modified carbon dioxide extraction—prediction of the extractability using molecular dynamic simulation M. Günther, M. Maus, K.G. Wagner, P.C. Schmidt
321
A simple predictive model for the tensile strength of binary tablets C.-Y. Wu, S.M. Best, A.C. Bentham, B.C. Hancock, W. Bonfield
331
Pharmacokinetic changes of DA-7867, a new oxazolidinone, after intravenous and oral administration to rats with short-term and long-term diabetes mellitus induced by streptozotocin S.K. Bae, S.H. Yang, S.J. Lee, J.W. Kwon, W.B. Kim, D.C. Lee, M.G. Lee
337
EUFEPS Announcemen
347
Calendar of Events
351
Vol. 25/4–5, July–August 2005 Research papers Comparative scale-up of three methods for producing ibuprofen-loaded nanoparticles S.A. Galindo-Rodríguez, F. Puel, S. Briançon, E. Allémann, E. Doelker, H. Fessi
357
The pharmacokinetics of pulmonary insulin in the in vitro isolated perfused rat lung: Implications of metabolism and regional deposition Y. Pang, M. Sakagami, P.R. Byron
369
Can protonated -blockers interact with biomembranes stronger than neutral isolipophilic compounds? A chromatographic study on three different phospholipid stationary phases (IAM-HPLC) F. Barbato, G. di Martino, L. Grumetto, M.I. La Rotonda
379
Salt formation in solid dispersions consisting of polyacrylic acid as a carrier and three basic model compounds resulting in very high glass transition temperatures and constant dissolution properties upon storage I. Weuts, D. Kempen, G. Verreck, J. Peeters, M. Brewster, N. Blaton, G. Van den Mooter
387
Optimisation of the predictive ability of artificial neural network (ANN) models: A comparison of three ANN programs and four classes of training algorithm A.P. Plumb, R.C. Rowe, P. York, M. Brown
395
Solid-state characterization of falicaine hydrochloride and isomorphic dyclonine hydrochloride. Part IV. Crystal polymorphism of local anaesthetic drugs A.C. Schmidt
407
A modification of the Hammett equation for predicting ionisation constants of p-vinyl phenols J. Sipilä, H. Nurmi, A.M. Kaukonen, J. Hirvonen, J. Taskinen, J. Yli-Kauhaluoma
417
Microencapsulated chitosan nanoparticles for lung protein delivery A. Grenha, B. Seijo, C. Remuñán-López
427
482
Contents, Volume 25 (2005) 479–482
Tissue penetration of cefpodoxime into the skeletal muscle and lung in rats P. Liu, R. Fuhrherr, A.I. Webb, B. Obermann, H. Derendorf
439
Enhanced oral paclitaxel absorption with vitamin E-TPGS: Effect on solubility and permeability in vitro, in situ and in vivo M.V.S. Varma, R. Panchagnula
445
Transport of nanoparticles across an in vitro model of the human intestinal follicle associated epithelium A. des Rieux, E.G.E. Ragnarsson, E. Gullberg, V. Préat, Y.-J. Schneider, P. Artursson
455
EUFEPS Announcements
467
Calendar of Events
471
Author Index Vol. 25
475
Contents Vol. 25
479
Contents, Volume 25 Vol. 25/1, May 2005 Review Microdialysis—theoretical background and recent implementation in applied life-sciences N. Plock, C. Kloft
1
Research papers Pharmacodynamic behaviour of the selective cyclooxygenase-2 inhibitor lumiracoxib in the lipopolysaccharidestimulated rat air pouch model R.E. Esser, R. Miserendino-Molteni, M. Sharr, X. Zhang, W. Porter, L. Ramos, J.A. Cramer, S. Zhuang, A. Georgieva, W. Maniara
25
Chitosan-reinforced alginate microspheres obtained through the emulsification/internal gelation technique A.J. Ribeiro, C. Silva, D. Ferreira, F. Veiga
31
Melt sonocrystallization of ibuprofen: Effect on crystal properties M. Manish, J. Harshal, P. Anant
41
Characterization of the 13-cis-retinoic acid/cyclodextrin inclusion complexes by phase solubility, photostability, physicochemical and computational analysis K.L. Yap, X. Liu, J.C. Thenmozhiyal, P.C. Ho
49
Vanillin suppresses in vitro invasion and in vivo metastasis of mouse breast cancer cells K. Lirdprapamongkol, H. Sakurai, N. Kawasaki, M.-K. Choo, Y. Saitoh, Y. Aozuka, P. Singhirunnusorn, S. Ruchirawat, J. Svasti, I. Saiki
57
A new sunscreen of the cinnamate class: Synthesis and enzymatic hydrolysis evaluation of glyceryl esters of p-methoxycinnamic acid Z.M.F. de Freitas, E.P. dos Santos, J.F. da Rocha, G.M. Dellamora-Ortiz, J.C.S. Gonçalves
67
Characterization of the rotating dialysis cell as an in vitro model potentially useful for simulation of the pharmacokinetic fate of intra-articularly administered drugs B.T. Pedersen, J. Østergaard, S.W. Larsen, C. Larsen
73
Atomic force microscopy and photon correlation spectroscopy: Two techniques for rapid characterization of liposomes B. Ruozi, G. Tosi, F. Forni, M. Fresta, M.A. Vandelli
81
Tissue distribution, pharmacokinetics and identification of roscovitine metabolites in rat M. Vita, M. Abdel-Rehim, S. Olofsson, Z. Hassan, L. Meurling, Å. Sidén, M. Sidén, T. Pettersson, M. Hassan
91
A solid-state NMR study of molecular mobility and phase separation in co-spray-dried protein–sugar particles E.J. Suihko, R.T. Forbes, D.C. Apperley
105
Permeability of pig urinary bladder wall: the effect of chitosan and the role of calcium M. Kerec, M. Bogataj, P. Veranicˇ , A. Mrhar
113
Estimation of dosing strategies aiming at maximizing utility or responder probability, using oxybutynin as an example drug S. Jönsson, M.O. Karlsson
123
doi:10.1016/S0928-0987(05)00185-5
480
Contents, Volume 25 (2005) 479–482
A comparative study of the potential of solid triglyceride nanostructures coated with chitosan or poly(ethylene glycol) as carriers for oral calcitonin delivery M. Garcia-Fuentes, C. Prego, D. Torres, M.J. Alonso
133
Pyrimidine and nucleoside -esters of L-Glu-Sar: Synthesis, stability and interaction with hPEPT1 A.H. Eriksson, P.L. Elm, M. Begtrup, B. Brodin, R. Nielsen, B. Steffansen
145
A simple method for differentiation of monoisotopic drug metabolites with hydrogen–deuterium exchange liquid chromatography/electrospray mass spectrometry A. Tolonen, M. Turpeinen, J. Uusitalo, O. Pelkonen
155
Pharmacokinetic–pharmacodynamic modelling of the schedule-dependent effect of the anti-cancer agent CHS 828 in a rat hollow fibre model L.E. Friberg, S.B. Hassan, E. Lindhagen, R. Larsson, M.O. Karlsson
163
EUFEPS Announcement
175
Calendar of Events
179
Instructions to Authors
183
Vol. 25/2–3, June 2005 Research papers Effect of experimental pH on the in vitro permeability in intact rabbit intestines and Caco-2 monolayer K.-J. Lee, N. Johnson, J. Castelo, P.J. Sinko, G. Grass, K. Holme, Y.-H. Lee
193
[99mTc]-hexakis-2-methoxyisobutyl
Biphasic accumulation kinetics of isonitrile in tumour cells and its modulation by lipophilic P-glycoprotein ligands T. Márián, L. Balkay, G. Szabó, Z.T. Krasznai, Z. Hernádi, L. Galuska, J. Szabó-Péli, O. Ésik, L. Trón, Z. Krasznai
201
pH-Dependent passive and active transport of acidic drugs across Caco-2 cell monolayers S. Neuhoff, A.-L. Ungell, I. Zamora, P. Artursson
211
Effect of staurosporine on N-glycosylation and cell adhesion to fibronectin of SW480 human colorectal adenocarcinoma cells T. Sato, M. Takahashi, T. Kawado, E. Takayama, K. Furukawa
221
AZD3582 increases heme oxygenase-1 expression and antioxidant activity in vascular endothelial and gastric mucosal cells G. Berndt, N. Grosser, J. Hoogstraate, H. Schröder
229
SDS-aided immobilization and controlled release of camptothecin from agarose hydrogel J. Liu, L. Li
237
QSAR analysis of substituted bis[(acridine-4-carboxamide)propyl]methylamines using optimized block-wise variable combination by particle swarm optimization for partial least squares modeling L. Lin, W.-Q. Lin, J.-H. Jiang, G.-L. Shen, R.-Q. Yu
245
Synthesis and antiamoebic activity of 3,7-dimethyl-pyrazolo[3,4-e][1,2,4] triazin-4-yl thiosemicarbazide derivatives S. Singh, K. Husain, F. Athar, A. Azam
255
Modulation of drug transport by selected flavonoids: Involvement of P-gp and OCT? M. Ofer, S. Wolffram, A. Koggel, H. Spahn-Langguth, P. Langguth
263
Acid–base properties of selected flavonoid glycosides C. Mielczarek
273
Polyelectrolyte complex formation and stability when mixing polyanions and polycations in salted media: A model study related to the case of body fluids T. Etrych, L. Leclercq, M. Boustta, M. Vert
281
Contents, Volume 25 (2005) 479–482
481
State of insulin self-association does not affect its absorption from the pulmonary route A. Hussain, F. Ahsan
289
Targeting liposomes with protein drugs to the blood–brain barrier in vitro C.C. Visser, S. Stevanovic´, L.H. Voorwinden, L. van Bloois, P.J. Gaillard, M. Danhof, D.J.A. Crommelin, A.G. de Boer
299
Investigation of the enhancing mechanism of sodium N-[8-(2-hydroxybenzoyl)amino]caprylate effect on the intestinal permeability of polar molecules utilizing a voltage clamp method S. Hess, V. Rotshild, A. Hoffman
307
Physical stability of the amorphous state of loperamide and two fragment molecules in solid dispersions with the polymers PVP-K30 and PVP-VA64 I. Weuts, D. Kempen, A. Decorte, G. Verreck, J. Peeters, M. Brewster, G. Van den Mooter
313
Hydrophilic solutes in modified carbon dioxide extraction—prediction of the extractability using molecular dynamic simulation M. Günther, M. Maus, K.G. Wagner, P.C. Schmidt
321
A simple predictive model for the tensile strength of binary tablets C.-Y. Wu, S.M. Best, A.C. Bentham, B.C. Hancock, W. Bonfield
331
Pharmacokinetic changes of DA-7867, a new oxazolidinone, after intravenous and oral administration to rats with short-term and long-term diabetes mellitus induced by streptozotocin S.K. Bae, S.H. Yang, S.J. Lee, J.W. Kwon, W.B. Kim, D.C. Lee, M.G. Lee
337
EUFEPS Announcemen
347
Calendar of Events
351
Vol. 25/4–5, July–August 2005 Research papers Comparative scale-up of three methods for producing ibuprofen-loaded nanoparticles S.A. Galindo-Rodríguez, F. Puel, S. Briançon, E. Allémann, E. Doelker, H. Fessi
357
The pharmacokinetics of pulmonary insulin in the in vitro isolated perfused rat lung: Implications of metabolism and regional deposition Y. Pang, M. Sakagami, P.R. Byron
369
Can protonated -blockers interact with biomembranes stronger than neutral isolipophilic compounds? A chromatographic study on three different phospholipid stationary phases (IAM-HPLC) F. Barbato, G. di Martino, L. Grumetto, M.I. La Rotonda
379
Salt formation in solid dispersions consisting of polyacrylic acid as a carrier and three basic model compounds resulting in very high glass transition temperatures and constant dissolution properties upon storage I. Weuts, D. Kempen, G. Verreck, J. Peeters, M. Brewster, N. Blaton, G. Van den Mooter
387
Optimisation of the predictive ability of artificial neural network (ANN) models: A comparison of three ANN programs and four classes of training algorithm A.P. Plumb, R.C. Rowe, P. York, M. Brown
395
Solid-state characterization of falicaine hydrochloride and isomorphic dyclonine hydrochloride. Part IV. Crystal polymorphism of local anaesthetic drugs A.C. Schmidt
407
A modification of the Hammett equation for predicting ionisation constants of p-vinyl phenols J. Sipilä, H. Nurmi, A.M. Kaukonen, J. Hirvonen, J. Taskinen, J. Yli-Kauhaluoma
417
Microencapsulated chitosan nanoparticles for lung protein delivery A. Grenha, B. Seijo, C. Remuñán-López
427
482
Contents, Volume 25 (2005) 479–482
Tissue penetration of cefpodoxime into the skeletal muscle and lung in rats P. Liu, R. Fuhrherr, A.I. Webb, B. Obermann, H. Derendorf
439
Enhanced oral paclitaxel absorption with vitamin E-TPGS: Effect on solubility and permeability in vitro, in situ and in vivo M.V.S. Varma, R. Panchagnula
445
Transport of nanoparticles across an in vitro model of the human intestinal follicle associated epithelium A. des Rieux, E.G.E. Ragnarsson, E. Gullberg, V. Préat, Y.-J. Schneider, P. Artursson
455
EUFEPS Announcements
467
Calendar of Events
471
Author Index Vol. 25
475
Contents Vol. 25
479